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Chemicals

GSK256066

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DESCRIPCIÓN

Supplier:Biorbyt
Reference:orb1301115
Name:GSK256066
Category:Chemicals
Subcategory:Small Molecules
Unit:1 mg
price :Consultar
note :801312-28-7
purity :99,66%
specificactivity :GSK256066 is a selective PDE4B(equal affinity to isoforms A-D) inhibitor with IC50 of 3.2 pM, > 380, 000-fold selectivity versus PDE1/2/3/5/6 and > 2500-fold selectivity against PDE4B versus PDE7.Phase 2.
Molecular weight :518,58


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